Cisapride

Cat. No.: OB0225WX-1573

Appearance: Solid

Purity: ≥99%

Identity: Confirmed by NMR, HPLC, and LC-MS.

Size:

INQUIRY Datasheet MSDS

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Product Overview

Description: Cisapride is a potent serotonin type 4 (5-HT4) receptor agonist that modulates gastrointestinal motility by stimulating receptors within the intestinal wall to enhance peristaltic action.

Synonym: Prepulsid; R 51619; Pridesia; Kaudalit; (±)-Cisaprid; Kinestase; 81098-60-4; Acenalin; Propulsin; 4-amino-5-chloro-N-[1-[3-(4-fluorophenoxy)propyl]-3-methoxypiperidin-4-yl]-2-methoxybenzamide; Risamal; 4-amino-5-chloro-N-{1-[3-(4-fluorophenoxy)propyl]-3-methoxypiperidin-4-yl}-2-methoxybenzamide; (+/-)-Cisapride; 4-amino-5-chloro-N-(1-(3-(4-fluorophenoxy)propyl)-3-methoxypiperidin-4-yl)-2-methoxybenzamide; 4-amino-5-chloro-N-[1-[3-(4-fluorophenoxy)propyl]-3-methoxy-4-piperidinyl]-2-methoxybenzamide; 4-Amino-5-Chloro-N-{1-[3-(4-Fluorophenoxy)Propyl]-3-Methoxy-4-Piperidinyl}-2-Methoxybenzamide; Benzamide, 4-amino-5-chloro-N-(1-(3-(4-fluorophenoxy)propyl)-3-methoxy-4-piperidinyl)-2-methoxy-, cis-; Benzamide, 4-amino-5-chloro-N-[1-[3-(4-fluorophenoxy)propyl]-3-methoxy-4-piperidinyl]-2-methoxy-, cis-; 4-amino-5-chloro-N-[1-{3-[(4-fluorophenyl)oxy]propyl}-3-(methyloxy)piperidin-4-yl]-2-(methyloxy)benzamide; 4-Amino-5-chloro-N-(1-[3-(4-fluorophenoxy)propyl]-3-methoxy-4-piperidinyl)-2-methoxybenzamide, cis- #

CAS No.: 81098-60-4

Compound CID: 2769

Formula: C₂₃H₂₉ClFN₃O₄

Formula Weight: 465.95

Specification

Targets&IC50: ERG channel (human): 9.4 nM; 5-HT4 receptor: 140 nM (EC50)

Relative Density: 1.29 g/cm³

Stability: 3 years in powder form.

Storage: Storage at -20°C.

Applications: Cisapride is used in gastrointestinal research as a prokinetic tool to study the activation of 5-HT4 receptors and the enhancement of acetylcholine release in the enteric nervous system.