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BGT226 maleate
Cat. No.:
OB0225LY-0390
Appearance:
Solid
Purity:
≥98%
Identity:
Confirmed by NMR and HPLC.
Size:
Add to basket
Product Overview
Description:
BGT226 maleate is an oral biologic drug that targets the PI3K/mTOR pathway and shows anti-cancer potential.
Synonym:
BGT226; NVP-BGT226 (maleate); NVP-BGT226; 1245537-68-1; (Z)-But-2-enedioic acid; 8-(6-methoxypyridin-3-yl)-3-methyl-1-[4-piperazin-1-yl-3-(trifluoromethyl)phenyl]imidazo[4,5-c]quinolin-2-one; 8-(6-methoxypyridin-3-yl)-3-methyl-1-(4-(piperazin-1-yl)-3-(trifluoromethyl)phenyl)-1H-imidazo[4,5-c]quinolin-2(3H)-one maleate; 8-(6-Methoxypyridin-3-yl)-3-methyl-1-(4-(piperazin-1-yl)-3-(trifluoromethyl)phenyl)-1,3-dihydro-2H-imidazo[4,5-c]quinolin-2-one maleate; 1-(3-(Trifluoromethyl)-4-(piperazin-1-yl)phenyl)-8-(6-methoxypyridin-3-yl)-3-methyl-1H-imidazo[4,5-c]quinolin-2(3H)-one maleic acid salt
CAS No.:
1245537-68-1
Compound CID:
57336745
Formula:
C28H25F3N6O2·C4H4O4
Formula Weight:
650.6
Specification
Stability:
3 years in powder form.
Storage:
Storage at -20°C.
Applications:
BGT226 maleate can be used for tumor biology research.
Library Information
Targets:
PI3K/Akt/mTOR pathway
Receptors:
mTOR; PI3Kα; PI3Kβ; PI3Kγ
Pathways:
Apoptosis; Autophagy; PI3K/Akt/mTOR signaling
Plate Number:
AOCL-6
Plate Location:
a5
Empty Location:
a1-h1; a12-h12
Container:
96-well plate
Formulation:
10 mM DMSO
DMSO Max Solubility:
60 mg/mL; 92.22 mM
Water Max Solubility:
<1 mg/mL (insoluble or slightly soluble)
Ethanol Max Solubility:
<1 mg/mL (insoluble or slightly soluble)
ALogP:
1.618
HBA_Count:
6
HBD_Count:
1
Rotatable Bond:
7





