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TGR5 receptor agonist
Cat. No.:
0225LY-0961
Appearance:
Solid
Purity:
≥99%
Identity:
Confirmed by NMR, and LC-MS.
Size:
Add to basket
Product Overview
Description:
TGR5 receptor agonist is a potent agonist specifically designed to target the TGR5 (GPCR19) receptor.
Synonym:
1197300-24-5; TGR5; CCDC; 3-(2-chlorophenyl)-N-(4-chlorophenyl)-N,5-dimethylisoxazole-4-carboxamide; 4-Isoxazolecarboxamide, 3-(2-chlorophenyl)-N-(4-chlorophenyl)-N,5-dimethyl-; 3-(2-chlorophenyl)-N-(4-chlorophenyl)-N,5-dimethyl-1,2-oxazole-4-carboxamide; MFCD17169972; 3-(2-chlorophenyl)-N-(4-chlorophenyl)-N,5-dimethyl-4-Isoxazolecarboxamide
CAS No.:
1197300-24-5
Compound CID:
44605616
Formula:
C18H14Cl2N2O2
Formula Weight:
361.22
Specification
Targets&IC50:
TGR5/GPCR19 (U2-OS cells): 6.8(pEC50); TGR5/GPCR19 (melanophore cells): 7.5(pEC50)
Relative Density:
1.346 g/cm3
Stability:
3 years in powder form.
Storage:
Storage at -20°C.
Applications:
TGR5 receptor agonist can be used in metabolic research to study the regulation of energy expenditure and glucose homeostasis.
Library Information
Target:
TGR5
Receptor:
TGR5
Pathways:
Protein kinase signaling
Plate Number:
AOCL-13
Plate Location:
d2
Empty Location:
a1-h1; a12-h12
Container:
96-well plate
Formulation:
10mM DMSO
DMSO Max Solubility:
50 mg/mL; 138.42 mM
Ethanol Max Solubility:
100 mM
