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CAY10650
Cat. No.:
OB0225WX-2085
Appearance:
Solid
Purity:
≥95%
Identity:
Confirmed by NMR, and HPLC.
Size:
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Product Overview
Description:
CAY10650 is a potent small molecule inhibitor of cytosolic phospholipase A2α (cPLA2α) characterized by an IC50 of 12 nM.
Synonym:
1233706-88-1; 3-isobutyryl-1-(2-oxo-3-(4-phenoxyphenoxy)propyl)-1H-indole-5-carboxylic acid; 1H-Indole-5-carboxylic acid,3-(2-methyl-1-oxopropyl)-1-[2-oxo-3-(4-phenoxyphenoxy)propyl]-
CAS No.:
1233706-88-1
Compound CID:
45102612
Formula:
C28H25NO6
Formula Weight:
471.5
Specification
Targets&IC50:
CPLA2α: 12 nM
Relative Density:
1.24 g/cm3
Stability:
3 years in powder form.
Storage:
Storage at -20°C.
Applications:
CAY10650 is utilized in inflammatory research as a potent inhibitor of cytosolic phospholipase A2 (cPLA2) to examine the reduction of arachidonic acid release and its effects on eicosanoid production.
Library Information
Target:
Phospholipase
Receptor:
cPLA2α
Pathways:
Metabolism
Plate Number:
AOCL-27
Plate Location:
f8
Empty Location:
a1-h1; a12-h12
Container:
96-well plate
Formulation:
10mM DMSO
DMSO Max Solubility:
40 mg/mL; 84.84 mM
