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Pristimerin
Cat. No.:
OB0225WX-2790
Appearance:
Solid
Purity:
≥99%
Identity:
Confirmed by NMR, and HPLC.
Size:
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Product Overview
Description:
Pristimerin is a natural triterpenoid that suppresses cancer cell proliferation (IC50: 0.2-4 micromolar) and reversibly inhibits monoacylglycerol lipase (MGL) with an IC50 of 93 nM.
Synonym:
1258-84-0
CAS No.:
1258-84-0
Formula:
C30H40O4
Formula Weight:
464.64
Specification
Stability:
3 years in powder form.
Storage:
Storage at -20°C.
Applications:
Pristimerin is used in oncology and signal transduction research as a triterpenoid quinone methide to investigate the inhibition of the proteasome and the suppression of NF-kappaB and STAT3 signaling in cancer cells.
Library Information
Target:
Lipase
Receptor:
MGL
Pathways:
Metabolism
Plate Number:
L6700-11
Empty Location:
a1-h1; a12-h12
Container:
96-well plate
Formulation:
10mM DMSO
DMSO Max Solubility:
12 mg/mL; 25.83 mM
ALogP:
5.7
HBA_Count:
3
HBD_Count:
1
Rotatable Bond:
2
