LY2608204

Cat. No.: OB0225WX-2468

Appearance: Solid

Purity: ≥99%

Identity: Confirmed by NMR, and HPLC.

Size:

INQUIRY Datasheet MSDS

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Product Overview

Description: LY2608204 is a potent small molecule activator of glucokinase (GK), exhibiting an effective concentration (EC50) of 42 nM.

Synonym: 1234703-40-2; LY-2608204; Globalagliatin; (1R,2S)-2-Cyclohexyl-1-(4-(cyclopropylsulfonyl)phenyl)-N-(5-((2-(1-pyrrolidinyl)ethyl)thio)-2-thiazolyl)cyclopropanecarboxamide; (1R,2S)-2-Cyclohexyl-1-(4-cyclopropylsulfonylphenyl)-N-[5-(2-pyrrolidin-1-ylethylsulfanyl)-1,3-thiazol-2-yl]cyclopropane-1-carboxamide; (1R,2S)-2-cyclohexyl-1-[4-(cyclopropanesulfonyl)phenyl]-N-(5-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-1,3-thiazol-2-yl)cyclopropane-1-carboxamide; Cyclopropanecarboxamide, 2-cyclohexyl-1-[4-(cyclopropylsulfonyl)phenyl]-N-[5-[[2-(1-pyrrolidinyl)ethyl]thio]-2-thiazolyl]-, (1R,2S)-; (1R,2S)-2-cyclohexyl-1-(4-(cyclopropanesulfonyl)phenyl)-N-(5-((2-(pyrrolidin-1-yl)ethyl)sulfanyl)-1,3-thiazol-2-yl)cyclopropane-1-carboxamide; MFCD21609257; (1R,2S)-2-Cyclohexyl-1-(4-(cyclopropylsulfonyl)phenyl)-N-(5-((2-(1-pyrrolidinyl)ethyl)sulfanyl)-1,3-thiazol-2-yl)cyclopropanecarboxamide; (1r,2s)-2-cyclohexyl-1-(4-cyclopropanesulfonyl-phenyl)-cyclopropanecarboxylic acid [5-(2-pyrrolidin-1-yl-ethylsulfanyl)-thiazol-2-yl]-amide

CAS No.: 1234703-40-2

Compound CID: 46832368

Formula: C₂₈H₃₇N₃O₃S₃

Formula Weight: 559.81

Specification

Stability: 3 years in powder form.

Storage: Storage at -20°C.

Applications: LY2608204 is used in metabolic research as a potent glucokinase activator to investigate the enhancement of glucose-stimulated insulin secretion and the regulation of hepatic glucose uptake.