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Vitamin B12 test kit

DGAT1-IN-1

Cat. No.: 0225LY-0723
Appearance: Solid
Purity: ≥99%
Identity: Confirmed by NMR, HPLC, and LC-MS.
Size:
DGAT1-IN-1
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Product Overview

Description: DGAT1-IN-1 is a high-potency inhibitor of diacylglycerol O-acyltransferase type 1 (DGAT1), featuring an IC50 value below 10 nM.
Synonym: 1449779-49-0; 2-(trans-4-(4-(2-((4-(Trifluoromethoxy)benzyl)carbamoyl)imidazo[1,2-a]pyridin-6-yl)phenyl)cyclohexyl)acetic acid; 2-[4-[4-[2-[[4-(trifluoromethoxy)phenyl]methylcarbamoyl]imidazo[1,2-a]pyridin-6-yl]phenyl]cyclohexyl]acetic acid; 2-((1r,4r)-4-(4-(2-((4-(trifluoromethoxy)benzyl)carbamoyl)imidazo[1,2-a]pyridin-6-yl)phenyl)cyclohexyl)acetic acid; (4-{4-[2-({[4-(trifluoromethoxy)phenyl]methyl}carbamoyl)imidazo[1,2-a]pyridin-6-yl]phenyl}cyclohexyl)acetic acid; Rel-2-((1r,4r)-4-(4-(2-((4-(Trifluoromethoxy)benzyl)carbamoyl)imidazo[1,2-a]pyridin-6-yl)phenyl)cyclohexyl)acetic acid
CAS No.: 1449779-49-0
Compound CID: 71696573
Formula: C30H28F3N3O4
Formula Weight: 551.56

Specification

Targets&IC50: DGAT-1: < 10 nM
Relative Density: 1.36 g/cm3
Stability: 3 years in powder form.
Storage: Storage at -20°C.
Applications: DGAT1-IN-1 can be used in preclinical metabolic studies to evaluate the role of DGAT1 in controlling intestinal fat absorption.

Library Information

Target: DGAT1
Receptor: DGAT1
Pathways: Metabolism
Plate Number: AOCL-10
Plate Location: c10
Empty Location: a1-h1; a12-h12
Container: 96-well plate
Formulation: 10mM DMSO
DMSO Max Solubility: 20 mg/mL; 36.26 mM
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