(E/Z)-GSK5182

Cat. No.: OB0225WX-1812

Appearance: Solid

Purity: ≥97%

Identity: Confirmed by NMR, HPLC, and LC-MS.

Size:

INQUIRY Datasheet MSDS

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Product Overview

Description: (E/Z)-GSK5182 is a racemic mixture of isomers functioning as a potent and selective inverse agonist for the estrogen-related receptor gamma (ERR-gamma) with an IC50 of 79 nM.

Synonym: GSK5182(Z/E); 2699724-40-6; GSK5182; GSK 5182; (Z)-4-(1-(4-(2-(dimethylamino)ethoxy)phenyl)-5-hydroxy-2-phenylpent-1-en-1-yl)phenol; 4-[(1Z)-1-{4-[2-(dimethylamino)ethoxy]phenyl}-5-hydroxy-2-phenylpent-1-en-1-yl]phenol; 4-[(Z)-1-[4-(2-dimethylaminoethoxy)phenyl]-5-hydroxy-2-phenylpent-1-enyl]phenol; 4-[(Z)-1-[4-[2-(dimethylamino)ethoxy]phenyl]-5-hydroxy-2-phenylpent-1-enyl]phenol; 4-[1-[4-[2-(dimethylamino)ethoxy]phenyl]-5-hydroxy-2-phenylpent-1-enyl]phenol; 4-(1-(4-(2-(Dimethylamino)ethoxy)phenyl)-5-hydroxy-2-phenylpent-1-en-1-yl)phenol; 4-[(z)-1-[4-(2-dimethylaminoethyloxy)phenyl]-hydroxy-2-phenylpent-1-enyl]phenol

CAS No.: 2699724-40-6

Compound CID: 6852176

Formula: C₂₇H₃₁NO₃

Formula Weight: 417.54

Specification

Stability: 3 years in powder form.

Storage: Storage at -20°C.

Applications: (E/Z)-GSK5182 is applied in endocrine and metabolic studies as a selective inverse agonist of the estrogen-related receptor gamma (ERR-gamma) to investigate the regulation of hepatic gluconeogenesis.