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Protein kinase G inhibitor-1
Cat. No.:
0225LY-1352
Appearance:
Solid
Purity:
≥98%
Identity:
Confirmed by NMR, and LC-MS.
Size:
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Product Overview
Description:
Protein kinase G inhibitor-1 functions as a high-potency antagonist of Protein kinase G, characterized by an IC50 value of 0.9 uM.
Synonym:
354544-70-0; 2-(Cyclopropanecarboxamido)-6-methyl-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxamide; 2-[(cyclopropylcarbonyl)amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide; 2-(cyclopropanecarbonylamino)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
CAS No.:
354544-70-0
Compound CID:
2862914
Formula:
C14H18N2O2S
Formula Weight:
278.37
Specification
Targets&IC50:
PKG: 0.9 uM
Stability:
3 years in powder form.
Storage:
Storage at -20°C.
Applications:
Protein kinase G inhibitor-1 can be used in signal transduction research to evaluate the effects of selective PKG blockade on vascular smooth muscle.
Library Information
Target:
PKA
Receptor:
PKA
Pathways:
cAMP signaling; GPCR/G protein signaling
Plate Number:
AOCL-18
Plate Location:
c10
Empty Location:
a1-h1; a12-h12
Container:
96-well plate
Formulation:
10mM DMSO
DMSO Max Solubility:
30 mg/mL; 107.77 mM
