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BQR-695
Cat. No.:
0225LY-0671
Appearance:
Solid
Purity:
≥99%
Identity:
Confirmed by NMR, and LC-MS.
Size:
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Product Overview
Description:
BQR-695 is a PI4K inhibitor showing IC50 values of 80 nM and 3.5 nM for human and Plasmodium PI4KIII-beta, respectively.
Synonym:
1513879-21-4; 2-((7-(3,4-dimethoxyphenyl)quinoxalin-2-yl)amino)-N-methylacetamide; N~2~-[7-(3,4-Dimethoxyphenyl)quinoxalin-2-Yl]-N-Methylglycinamide
CAS No.:
1513879-21-4
Compound CID:
112499905
Formula:
C19H20N4O3
Formula Weight:
352.39
Specification
Targets&IC50:
P. falciparum (PI4KIIIβ): 3.5 nM; PI4KIIIβ (human): 80 nM
Relative Density:
1.250 g/cm3
Stability:
3 years in powder form.
Storage:
Storage at -20°C.
Applications:
BQR-695 can be used in drug discovery to investigate the selective targeting of phosphatidylinositol kinases.
Library Information
Target:
PI4K; PI3K; Parasite protein
Receptor:
PI3KIIIβ; PI4K
Pathways:
Microbiology/Virology; PI3K/Akt/mTOR signaling
Plate Number:
AOCL-9
Plate Location:
f8
Empty Location:
a1-h1; a12-h12
Container:
96-well plate
Formulation:
10mM DMSO
DMSO Max Solubility:
50 mg/mL; 141.89 mM
