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DG172 dihydrochloride
Cat. No.:
0225LY-0814
Appearance:
Solid
Purity:
≥99%
Identity:
Confirmed by NMR, and LC-MS.
Size:
Add to basket
Product Overview
Description:
DG172 dihydrochloride serves as an antagonist of the PPAR beta/delta receptor, with an IC50 of 27 nM.
Synonym:
DG172 (dihydrochloride); DG-172 dihydrochloride; 1361504-77-9; DG-172 dihydrochloride; (Z)-2-(2-bromophenyl)-3-(4-(4-methylpiperazin-1-yl)phenyl)acrylonitrile dihydrochloride; (Z)-2-(2-bromophenyl)-3-[4-(4-methylpiperazin-1-yl)phenyl]prop-2-enenitrile;dihydrochloride
CAS No.:
1361504-77-9
Compound CID:
57342888
Formula:
C20H22BrCl2N3
Formula Weight:
455.2
Specification
Targets&IC50:
PPARβ/δ: 27 nM
Stability:
3 years in powder form.
Storage:
Storage at -20°C.
Applications:
DG172 dihydrochloride can be used in nuclear receptor research to study the selective antagonism of PPAR beta/delta.
Library Information
Target:
PPAR
Receptor:
PPAR
Pathways:
Metabolism; DNA damage/DNA repair
Plate Number:
AOCL-11
Plate Location:
e3
Empty Location:
a1-h1; a12-h12
Container:
96-well plate
Formulation:
10mM DMSO
DMSO Max Solubility:
14.29 mg/mL; 31.39 mM
