Products
Online Inquiry

Please note that we are not a pharmacy or clinic, so we are unable to see patients and do not offer diagnostic and treatment services for individuals.

Vitamin B12 test kit

XMD16-5

Cat. No.: 0225LY-0880
Appearance: Solid
Purity: ≥99%
Identity: Confirmed by NMR, HPLC, and LC-MS.
Size:
XMD16-5
Add to basket

Product Overview

Description: XMD16-5 is an inhibitor of TNK2, a protein whose genomic amplification and disrupted signaling are linked to metastasis and late-stage progression in breast, prostate, lung, and gastrointestinal cancers.
Synonym: 1345098-78-3; 2-[4-(4-hydroxypiperidin-1-yl)anilino]-11-methyl-5H-pyrimido[4,5-b][1,4]benzodiazepin-6-one; Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 18; 2-((4-(4-hydroxypiperidin-1-yl)phenyl)amino)-11-methyl-5,11-dihydro-6H-benzo[e]pyrimido[5,4-b][1,4]diazepin-6-one; 2-((4-(4-hydroxypiperidin-1-yl)phenyl)amino)-11-methyl-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one; 3-[4-(4-Hydroxy-piperidin-1-yl)-phenylamino]-5-methyl-5,11-dihydro-2,4,5,11-tetraaza-dibenzo[a,d]cyclohepten-10-one; 5-{[4-(4-hydroxypiperidin-1-yl)phenyl]amino}-2-methyl-2,4,6,9-tetraazatricyclo[9.4.0.0(3),?]pentadeca-1(15),3,5,7,11,13-hexaen-10-one
CAS No.: 1345098-78-3
Compound CID: 57340666
Formula: C23H24N6O2
Formula Weight: 416.48

Specification

Targets&IC50: R806Q: 77 nM; D163E: 16nM
Relative Density: 1.347 g/cm3
Stability: 3 years in powder form.
Storage: Storage at -20°C.
Applications: XMD16-5 can be used in kinase signaling research to study the dual inhibition of BRK and ERK5.

Library Information

Target: Tyrosinase; PPAR
Receptor: TNK2; Tyrosinase
Pathways: Proteases/Proteasome; DNA damage/DNA repair; Metabolism
Plate Number: AOCL-12
Plate Location: c9
Empty Location: a1-h1; a12-h12
Container: 96-well plate
Formulation: 10mM DMSO
DMSO Max Solubility: 45 mg/mL; 108.05 mM
Water Max Solubility: <1 mg/mL (insoluble or slightly soluble)
Ethanol Max Solubility: 5 mg/mL; 12.01 mM
Inquiry
0
Inquiry Basket

Copyright © Protheragen. All rights reserves.