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Rabusertib
Cat. No.:
OB0225LY-0392
Appearance:
Solid
Purity:
≥99%
Identity:
Confirmed by NMR and HPLC.
Size:
Add to basket
Product Overview
Description:
Rabusertib is a small molecule drug that acts primarily as a protein kinase inhibitor, targeting the proliferation and survival signaling pathways of tumor cells.
Synonym:
911222-45-2; (S)-1-(5-Bromo-4-methyl-2-(morpholin-2-ylmethoxy)phenyl)-3-(5-methylpyrazin-2-yl)urea; 1-[5-Bromo-4-methyl-2-[[(2S)-morpholin-2-yl]methoxy]phenyl]-3-(5-methylpyrazin-2-yl)urea; Urea, N-(5-bromo-4-methyl-2-((2S)-2-morpholinylmethoxy)phenyl)-N'-(5-methyl-2- pyrazinyl)-; (N-(5-bromo-4-methyl-2-{[(2S)-morpholin-2-yl]methoxy}phenyl)-N'-(5-methylpyrazin-2-yl)urea
CAS No.:
911222-45-2
Compound CID:
11955855
Formula:
C18H22BrN5O3
Formula Weight:
436.3
Specification
Relative Density:
1.461 g/cm3
Stability:
3 years in powder form.
Storage:
Storage at -20°C.
Applications:
Rabusertib can be used in tumor biology research to help understand the mechanisms of cell proliferation and the effects on specific signaling pathways.
Library Information
Targets:
Chk; PDK
Receptors:
Chk1; PDK1
Pathways:
PI3K/Akt/mTOR signaling; Autophagy; Cell cycle/Checkpoint
Plate Number:
AOCL-6
Plate Location:
a7
Empty Location:
a1-h1; a12-h12
Container:
96-well plate
Formulation:
10 mM DMSO
DMSO Max Solubility:
4.36 mg/mL; 10 mM
Water Max Solubility:
<1 mg/mL (insoluble or slightly soluble)
Ethanol Max Solubility:
<1 mg/mL (insoluble or slightly soluble)
