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Phentolamine mesylate
Cat. No.:
0225LY-1221
Appearance:
Solid
Purity:
≥99%
Identity:
Confirmed by NMR, and LC-MS.
Size:
Add to basket
Product Overview
Description:
Phentolamine mesylate is a nonselective alpha-adrenergic antagonist used for treating hypertensive emergencies, pheochromocytoma, Raynaud's disease, and various peripheral vascular conditions.
Synonym:
Phentolamine methanesulfonate; Phentolamine mesilate; 65-28-1; Phentolamine (mesylate); OraVerse; Regitine mesylate; Phentolamine methanesulfonate salt; Regitin methanesulphonate; Regitine methanesulfonate; Mesylate phentolamine; Phentolamine methanesulphonate; 3-(((4,5-dihydro-1H-imidazol-2-yl)methyl)(p-tolyl)amino)phenol methanesulfonate; Phenol,3-[[(4,5-dihydro-1H-imidazol-2-yl)methyl](4-methylphenyl)amino]-,monomethanesulfonate (salt); m-(N-(2-Imidazolin-2-ylmethyl)-p-toluidino)phenol monomethanesulfonate (salt); Phenol, 3-(((4,5-dihydro-1H-imidazol-2-yl)methyl)(4-methylphenyl)amino)-, monomethanesulfonate (salt)
CAS No.:
65-28-1
Compound CID:
91430
Formula:
C17H19N3O·CH4O3S
Formula Weight:
377.46
Specification
Targets&IC50:
α-adrenoceptor: 5 - 30 nM
Relative Density:
1.2256 g/cm3
Stability:
3 years in powder form.
Storage:
Storage at -20°C.
Applications:
Phentolamine mesylate can be used in pharmacological research to investigate the reversible blockade of both alpha-1 and alpha-2 adrenergic receptors.
Library Information
Target:
α-Adrenergic receptor
Receptor:
GPCR
Pathways:
Neuronal signaling; GPCR/G protein signaling
Plate Number:
AOCL-16
Plate Location:
f8
Empty Location:
a1-h1; a12-h12
Container:
96-well plate
Formulation:
10mM DMSO
DMSO Max Solubility:
60 mg/mL; 158.96 mM
Water Max Solubility:
37.8 mg/mL; 100.14 mM





